Therapeutic index number full#

Receptor that does not bind drug when the drug concentration is sufficient to produce maximal effect present when K d > EC 50Д¬omponent of a system that accomplishes the biologic effect after the receptor is activated by an agonist often a channel or enzyme molecule, may be part of the receptor moleculeДЄ drug that activates its receptor upon bindingДЄ drug that binds without activating its receptor and thereby prevents activation by an agonistДЄ pharmacologic antagonist that can be overcome by increasing the concentration of agonistДЄ pharmacologic antagonist that cannot be overcome by increasing agonist concentrationДЄ drug that counters the effects of another by binding to a different receptor and causing opposing effectsДЄ drug that counters the effects of another by binding the agonist drug (not the receptor)ДЄ drug that binds to a receptor molecule without interfering with normal agonist binding but alters the response to the normal agonistДЄ drug that binds to its receptor but produces a smaller effect at full dosage than a full agonistДЄ drug that binds to the inactive state of receptor molecules and decreases constitutive activity (see text)ДЄ graph of increasing response to increasing drug concentration or doseДЄ graph of the fraction of a population that shows a specified response at progressively increasing doses Baidyanath is Indias most trusted brand for Ayurvedic treatment.

Specific region of the receptor molecule to which the drug binds The therapeutic index of the benzodiazepines is high and the mortality rate associated with poisoning due. A molecule to which a drug binds to bring about a change in function of the biologic systemДЄ molecule to which a drug may bind without changing any function